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Description

Abilify is prescribed for:

  • Major depressive disorder (adjunct treatment)
  • Schizophrenia in adults/adolescents
  • Bipolar disorder (manic/mixed episodes)
  • Irritability associated with autism in pediatric patients

Mechanism of Action

  • Partial agonist at D2 and 5-HT1A receptors
  • Antagonist at 5-HT2A receptors
  • Moderate affinity for histamine/alpha-adrenergic receptors

Dosage & Administration

  • Initial dose: 10-15mg once daily
  • May be adjusted based on response
  • Can be taken with/without food

Important Safety Information

Contraindications:

  • Hypersensitivity to aripiprazole
  • Breastfeeding

Precautions:

  • Increased suicide risk in young patients
  • Not for dementia-related psychosis in elderly
  • May impair judgment/motor skills
  • Risk of hyperglycemia (monitor blood sugar)
  • Avoid alcohol and overheating

Potential Side Effects

Common:

  • Nausea/constipation
  • Headache/dizziness
  • Insomnia/restlessness
  • Weight gain

Serious (seek medical help):

  • Neuroleptic malignant syndrome
  • Tardive dyskinesia
  • Stroke risk
  • Uncontrolled movements

Drug Interactions

Levels decreased by:

  • Carbamazepine
  • Phenytoin
  • Rifampin

Levels increased by:

  • Ketoconazole/other antifungals
  • Fluoxetine/paroxetine
  • Quinidine

Missed Dose/Overdose

  • Missed dose: Take when remembered (skip if near next dose)
  • Overdose symptoms: Vomiting, tremors, cardiac abnormalities

Storage Instructions

  • Keep at room temperature
  • Store in original container
  • Protect from moisture

Note: Regular monitoring required for glucose levels and neurological symptoms. Report any unusual movements or mood changes to your doctor immediately.

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